Timolol yog ib qho kev kho mob kws kho mob tsis haum xeeb, uas yog ntawm cov tshuaj tseem ceeb thiab tseem ceeb heev. Xav txog cov ntaub ntawv tseem ceeb ntawm cov tee rau lub qhov muag ntawm Timolol, uas tus neeg mob xav tau thaum siv cov tshuaj no.
Teeb thiab daim ntawv ntawm Timolol npaj
Raws li txoj cai, qhov muag tshuaj ntawm Timolol muaj nyob rau hauv cov yas hwj-dej. Lub active feem ntawm cov tshuaj yog timolol nyob rau hauv daim ntawv ntawm maleate (txiv hmab txiv ntoo acidic ntsev). Cov ntsiab lus ntawm cov dej cawv nyob rau hauv cov qhov muag yuav tau 0.5% (5 mg timolol hauv 1 ml kua) los yog 0.25% (2.5 mg timolol hauv 1 ml kua).
Additives rau qhov muag tee timolol:
- sodium chloride;
- benzalkonium chloride;
- sodium dihydrogen phosphate dihydrate;
- disodium phosphate dodecahydrate;
- sodium edetate;
- distilled dej.
Cov kev qhia rau kev siv cov tshuaj tsuag Timolol:
- ocular hypertension (nce siab hauv siab);
- ntev qhib - lub kaum ntse ntse glaucoma ;
- Closed-glut glaucoma (nrog meotics);
- lwm yam glaucoma (uveal, posttraumatic, aphakic);
- Congenital glaucoma (nrog rau kev ua tsis zoo ntawm lwm cov kev ntsuas).
Pharmacological kev txiav txim ntawm qhov muag tshuaj Timolol
Cov khoom tseem ceeb ntawm cov tshuaj no yog ib yam ua tau zoo heev, tsis yog cov khoom siv beta-adrenergic reseptor blocker (ib qho cuab yeej uas ua rau kev tuav cov hlab ntsha tsis zoo).
Cov nyhuv ntawm cov tshuaj yog vim yog vim muaj kev txo qis ntawm cov kua hauv lub hauv siab, tab sis qee qhov kev nce hauv kev tawm mus tsis raug cais tawm. Ncos ntawm cov roj hmab tsis cuam tshuam qhov loj me ntawm tub ntxhais kawm, kev pab thiab kev tawg, thiab tseem cia saib xyuas cov mob hauv siab (ophthalmotonus) thaum pw tsaug zog.
Txo cov kev mob ntawm ophthalmotonus yog ua tiav ob qho tibsi nrog cov pib ua ntej thiab nrog rau kev mob siab nyob hauv nruab siab. Cov nyhuv yog pom, raws li txoj cai, 20 feeb tom qab thov kev siv tshuaj, nce mus txog qhov siab tshaj 1 mus rau 2 xuab moos. Lub sij hawm ntawm kev txiav txim ntawm dauv ntawm timolol yog txog 24 xuab moos.
Timolol maleate yog ntxaum ntxaum los ntawm lub pob kws. Hauv ib qho me me, cov tshuaj nkag mus rau hauv cov kev ua pa los ntawm kev nqus ntawm cov hlab ntsha ntawm cov kabmob sib kis thiab cov kua muag tawm.
Txoj kev ntawm kev tswj hwm thiab hom kev noj tshuaj timolol
Raws li cov lus qhia rau kev siv ntawm lub qhov muag tshuaj Timolol, cov tshuaj yog siv ib qho kev tov txhua 1-2 zaug ntawm ib hnub nyob hauv qis lub qhov muag ntawm lub qhov muag. Qhov tshuaj ntawm qhov kev daws cov tshuaj no yog kev pom zoo los ntawm tus kws kho mob ib tus zuj zus. Yog tias tsis muaj txig txaus, koj yuav tsum pib siv cov tshuaj kom ntau. Tom qab tswj kev tawm hauv lub siab, cov tshuaj ntawm qhov tshuaj poob rau 1 poob ib hnub ib zaug.
Cov tshuaj yog npaj rau kev siv mus ntev (ntawm qhov nruab nrab, mus txog 6 lub lim tiam). Lub sij hawm ntawm kev kho mob nyob ntawm cov kab mob ntawm cov kab mob. Kev so hauv kev siv cov tshuaj ntawm cov roj ntoos timolol los yog cov kev hloov ntawm cov tshuaj yuav tsum tau nqa tawm tsuas yog thaum pom zoo los ntawm tus kws kho mob.
Tej Teebmeem ntawm Timolol Ncoog:
- txo ntawm lacrimation;
- mob khaub thuas hnoos hawb pob;
- taw tes nto keratopathy;
- Cov tsos mob ntawm cov tsos mob me me.
Hauv qee cov neeg mob uas siv lub tshuaj ntev heev, cov kev mob tshwm sim muaj peev xwm:
- arrhythmia;
- bradycardia;
- kev mob hypotension;
- txog kev ua tsis taus pa ;
- bronchospasm;
- kiv taub hau.
Contraindications rau kev siv cov tee Timolol:
- bronchial hawb pob;
- tus kab mob ntev obstructive pulmonary;
- sinus bradycardia;
- atrioventricular blockade ntawm II thiab III degree;
- ntshav qab zib mellitus;
- lub plawv tsis ua haujlwm;
- cev xeeb tub thiab lactation;
- hypersensitivity rau lub Cheebtsam ntawm yeeb tshuaj.
Timolol - analogues
Timolol nyob hauv kev sib tham nrog ib tus kws kho mob tuaj yeem hloov nrog cov tshuaj uas muaj kev zoo xws li cov tshuaj pharmacological. Cov no suav nrog:
- Tiv thaiv;
- Fotil;
- Nyeem;
- Xalatan;
- Pilocarpine;
- Betoptik.